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Bisindolylmaleimide VIII acetate
CAS No. 138516-31-1
Bisindolylmaleimide VIII acetate ( Ro 31-7549 acetate; Bis VIII acetate )
产品货号. M23542 CAS No. 138516-31-1
Bisindolylmaleimide VIII acetate is a potent and selective PKC inhibitor (IC50: 158 nM for rat brain PKC).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥1272 | 有现货 |
|
| 10MG | ￥2017 | 有现货 |
|
| 25MG | ￥4236 | 有现货 |
|
| 50MG | ￥6148 | 有现货 |
|
| 100MG | ￥8586 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Bisindolylmaleimide VIII acetate
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Bisindolylmaleimide VIII acetate is a potent and selective PKC inhibitor (IC50: 158 nM for rat brain PKC).
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产品描述Bisindolylmaleimide VIII acetate is a potent and selective PKC inhibitor (IC50: 158 nM for rat brain PKC). It has IC50s of 53, 195, 163, 213, and 175 nM for PKC-α, PKC-βI, PKC-βII, PKC-γ, PKC-ε, respectively.
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同义词Ro 31-7549 acetate; Bis VIII acetate
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通路Apoptosis
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靶点Apoptosis
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受体Apoptosis;PKC;PKCα;PKCβ1;PKCβ2;PKCγ;PKCε
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研究领域——
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适应症——
化学信息
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CAS Number138516-31-1
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分子量458.5
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分子式C26H26N4O4
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纯度>98% (HPLC)
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溶解度——
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SMILESO=C(C(C1=CN(CCCN)C2=C1C=CC=C2)=C3C4=CN(C)C5=C4C=CC=C5)NC3=O.CC(O)=O
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Wilkinson SE, et al. Isoenzyme specificity of bisindolylmaleimides, selective inhibitors of protein kinase C. Biochem J. 1993 Sep 1;294 ( Pt 2):335-7.
产品手册
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